Drug Repurposing Data Package
This package has 13 modules. The Drug-Protein Relationships and Drug Targets Module has 4 tables. Preview the first five rows of each table or Explore the schema
Drug-Protein Relationships and Drug Targets Module
4 Tables
Describes the relationship between drugs and targets, enzymes, carriers, or transporters. Annotation includes the pharmacological action, and the type of interaction (antagonist, agonist, substrate, inhibitor, or inducer).
biodb_id | name | kind | organism | drug_targets |
|---|---|---|---|---|
BE0000001 | Peptidoglycan D,D-transpeptidase FtsI | protein | Haemophilus influenzae (strain ATCC 51907 / DSM 11121 / KW20 / Rd) | 0 |
BE0000002 | Histidine decarboxylase | protein | Humans | 0 |
BE0000003 | Glutaminase liver isoform, mitochondrial | protein | Humans | 0 |
BE0000004 | Coagulation factor XIII A chain | protein | Humans | 0 |
BE0000005 | Nitric oxide synthase, inducible | protein | Humans | 0 |
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biodb_id | component_type | component_id |
|---|---|---|
BE0000001 | Polypeptide | P45059 |
BE0000002 | Polypeptide | P19113 |
BE0000003 | Polypeptide | Q9UI32 |
BE0000004 | Polypeptide | P00488 |
BE0000005 | Polypeptide | P35228 |
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id | type | drug_id | biodb_id | pdb_id | position | pharmacological_action | antagonist | agonist | substrate | inhibitor | inducer | other_action | inducer_strength | inhibitor_strength | induction_clinically_sig | inhibition_clinically_sig |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
1 | TargetBond | 1 | BE0000048 | 1 | yes | 0 | 0 | 0 | 1 | 0 | unknown | 0 | 0 | |||
2 | TargetBond | 2 | BE0000767 | 1 | yes | 0 | 0 | 0 | 0 | 0 | binder | 0 | 0 | |||
3 | TargetBond | 4 | BE0000658 | 1 | yes | 0 | 0 | 0 | 0 | 0 | ligand | 0 | 0 | |||
4 | TargetBond | 5 | BE0000704 | 1 | yes | 0 | 0 | 0 | 1 | 0 | antibody | unknown | 0 | 0 | ||
5 | TargetBond | 6 | BE0000048 | 1 | yes | 0 | 0 | 0 | 1 | 0 | unknown | 0 | 0 |
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uniprot_id | name | uniprot_name | gene_name | organism_id | molecular_weight | theoretical_pi | general_function | specific_function | signal_regions | transmembrane_regions | pdb_ids | genbank_gene_id | genbank_protein_id | genecard_id | locus | genatlas_id | hgnc_id | meta_cyc_id | ncbi_sequence_ids | tissue_specificity | cofactor | subunit | cellular_location | amino_acid_sequence | gene_sequence |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
A0A023W3H0 | OXA-48 carbapenemase | A0A023W3H0_KLEPN | OXA-48 | 144 | 16920.07 | penicillin binding | >lcl|BSEQ0022471|Class D OXA-48 carbapenemase
VVKDEHQVFKWDGQTRDIATWNRDHNLITAMKYSVVPVYQEFARQIGEARMSKMLHAFDY
GNEDISGNVDSFWLDGGIRISATEQISFLRKLYHNKLHVSERSQRIVKQAMLTEANGDYI
IRAKTGYSTRIEPKIGWWVGWVELD | ||||||||||||||||||
A0A024R1R8 | Translation machinery-associated protein 7B | TMA7B_HUMAN | TMA7B | 154 | 7091.405 | TMA7B | 22q13.1 | HGNC:53893 | >lcl|BSEQ0069905|Translation machinery-associated protein 7B
MSSHEGGKKKALKQPKKQAKEMDEEEKAFKQKQKEEQKKLEVLKAKVVGKGPLATGGIKK
SGKK | ||||||||||||||||
A0A024RBG1 | Diphosphoinositol polyphosphate phosphohydrolase NUDT4B | NUD4B_HUMAN | NUDT4B | 154 | 20434.03 | Cleaves a beta-phosphate from the diphosphate groups in PP-InsP5 (diphosphoinositol pentakisphosphate), PP-InsP4 and [PP]2-InsP4 (bisdiphosphoinositol tetrakisphosphate), suggesting that it may play a role in signal transduction. Also able to catalyze the hydrolysis of dinucleoside oligophosphate Ap6A, but not Ap5A. The major reaction products are ADP and p4a from Ap6A. Also able to hydrolyze 5-phosphoribose 1-diphosphate. Does not play a role in U8 snoRNA decapping activity. Binds U8 snoRNA | bis(5'-adenosyl)-hexaphosphatase activity | NUDT4B | 1q21.2 | HGNC:18012 | Cytoplasm | >lcl|BSEQ0064393|Diphosphoinositol polyphosphate phosphohydrolase NUDT4B
MMKFKPNQTRTYDREGFKKRAACLCFRSEQEDEVLLVSSSRYPDQWIVPGGGMEPEEEPG
GAAVREVYEEAGVKGKLGRLLGIFEQNQDRKHRTYVYVLTVTEILEDWEDSVNIGRKREW
FKVEDAIKVLQCHKPVHAEYLEKLKLGCSPANGNSTVPSLPDNNALFVTAAQTSGLPSSV
R | |||||||||||||
A0A059JJ46 | ABC multidrug transporter MDR2 | MDR2_TRIIM | MDR2 | 1913 | 145278.17 | Pleiotropic ABC efflux transporter that may be involved in the modulation susceptibility to a wide range of unrelated cytotoxic compounds, including terbinafine, 4-nitroquinoline N-oxide, and ethidium bromide (PubMed:16849730). May play a role in pathogenicity (PubMed:19141731). | ABC-type transporter activity | 93-113
147-167
219-239
242-262
325-345
358-378
762-782
810-830
884-904
910-930
995-1015
1025-1045 | Cell membrane | >lcl|BSEQ0052180|ABC multidrug transporter MDR2
MVEVSEKPNTQDDGVSKQENRNPASSSSSTSDKEKVAKKGNSDATKSSTPEDLDAQLAHL
PEHEREILKQQLFIPDAKATYGTLFRYATRNDMIFLAIVSLASIAAGAALPLFTVLFGSL
AGTFRDIALHRITYDEFNSILTRNSLYFVYLGIAQFILLYVSTVGFIYVGEHITQKIRAK
YLHAILRQNIGFFDKLGAGEVTTRITADTNLIQDGISEKVGLTLTALSTFFSAFIIGYVR
YWKLALICSSTIVAMILVMGGISRFVVKSGRMTLVSYGEGGTVAEEVISSIRNATAFGTQ
EKLARQYEVHLKEARKWGRRLQMMLGIMFGSMMAIMYSNYGLGFWMGSRFLVGGETDLSA
IVNILLAIVIGSFSIGNVAPNTQAFASAISAGAKIFSTIDRVSAIDPGSDEGDTIENVEG
TIEFRGIKHIYPSRPEVVVMEDINLVVPKGKTTALVGPSGSGKSTVVGLLERFYNPVSGS
VLLDGRDIKTLNLRWLRQQISLVSQEPTLFGTTIFENIRLGLIGSPMENESEEQIKERIV
SAAKEANAHDFIMGLPDGYATDVGQRGFLLSGGQKQRIAIARAIVSDPKILLLDEATSAL
DTKSEGVVQAALDAASRGRTTIVIAHRLSTIKSADNIVVIVGGRIAEQGTHDELVDKKGT
YLQLVEAQKINEERGEESEDEAVLEKEKEISRQISVPAKSVNSGKYPDEDVEANLGRIDT
KKSLSSVILSQKRSQEKETEYSLGTLIRFIAGFNKPERLIMLCGFFFAVLSGAGQPVQSV
FFAKGITTLSLPPSLYGKLREDANFWSLMFLMLGLVQLVTQSAQGVIFAICSESLIYRAR
SKSFRAMLRQDIAFFDLPENSTGALTSFLSTETKHLSGVSGATLGTILMVSTTLIVALTV
ALAFGWKLALVCISTVPVLLLCGFYRFWILAQFQTRAKKAYESSASYACEATSSIRTVAS
LTREQGVMEIYEGQLNDQAKKSLRSVAKSSLLYAASQSFSFFCLALGFWYGGGLLGKGEY
NAFQFFLCISCVIFGSQSAGIVFSFSPDMGKAKSAAADFKRLFDRVPTIDIESPDGEKLE
TVEGTIEFRDVHFRYPTRPEQPVLRGLNLTVKPGQYIALVGPSGCGKSTTIALVERFYDT
LSGGVYIDGKDISRLNVNSYRSHLALVSQEPTLYQGTIRDNVLLGVDRDDVPDEQVFAAC
KAANIYDFIMSLPDGFGTVVGSKGSMLSGGQKQRIAIARALIRDPKVLLLDEATSALDSE
SEKVVQAALDAAAKGRTTIAVAHRLSTIQKADIIYVFDQGRIVESGTHHELLQNKGRYYE
LVHMQSLEKTQ | |||||||||||||||
A0A068JFB7 | Beta-lactamase SHV | A0A068JFB7_ECOLX | blaSHV | 90 | 14354.285 | beta-lactamase activity | >lcl|BSEQ0052113|Beta-lactamase
GLTAFLRQIGDNVTRLDRWETELNEALPGDARDTTTPASMAATLRKLLTSQRLSARSQRQ
LLQWMVDDRVAGPLIRSVLPAGWFIADKTGASKRGARGIVALLGPNNKAERIVVIYLRDT
PASMAERNQQ |
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